FLT3

Receptor-type tyrosine-protein kinase FLT3

3 Targeting Drugs
5 Resistance Mutations
6JQR Structure Loaded
3D Structure PDB: 6JQR
Switch structure: RCSB ↗
Protein Information
UniProt Accession P36888 ↗
Gene Name FLT3
Cellular Location Membrane
General Function Vascular endothelial growth factor-activated receptor activity
Resistance Mutations Across All Drugs
Mutation Drug Source Resistance Samples
p.D835Y Sorafenib COSMIC 12
p.D835H Sorafenib COSMIC 12
p.D835X Sorafenib COSMIC 12
p.F691L Sorafenib COSMIC 12
p.D835Y Sunitinib COSMIC 9